Description

Trenbolone Acetate Landerlan

75mg/ml.

Injectable Oily Solution

Deep intramuscular route

Formula:

Each ml of solution for injection contains:
Trenbolone Acetate…………………………………………75mg
Excipients……………………………………………….…… q.s.

Content 10ml.

Mechanism of action

TREMBOLONE is a strong androgen that lacks estrogenic activity.
Structurally, TREMBOLONE is a 19 nor steroid, derived from nandrolone. The double bonds at C9 and C11 make TREMBOLONE very different in appearance than its relative nandrolone.
Its estrogenic activity has been eliminated. This is the result of the C9-10 double bond. This bond does not seem to be able to be removed metabolically, which is the only possible way for this compound to convert to estrogen. Although nandrolone is rarely thought of as an estrogenic steroid, conversion to estradiol is still possible to some extent. Therefore, the fact that TREMBOLONE does not convert to estradiol remains a significant difference between the two steroids. The androgenic activity of TREMBOLONE is also much stronger than that of its relative, nandrolone. This is due to two interesting traits: first, TREMBOLONE does not appear to promote 5-alpha reduction in humans. As such, it does not exhibit strong anabolic-androgenic dissociation like nandrolone, making it much more androgenic. Furthermore, induction of the double bond at C9 and C11 appears to increase binding to androgen receptors. This represents a second way in which the potency of TREMBOLONE is increased.
TREMBOLONE also suppresses natural testosterone production rapidly, this may necessitate the use of a testosterone-stimulating drug in order to avoid a steep drop when use is discontinued. Although listed as a "non-progestational" steroid in the literature, several studies clearly show that TREMBOLONE binds to these receptors. As we know all sex steroids promote negative feedback inhibition of testosterone production.

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